F2RL1
F2R like trypsin receptor 1
- Ensembl:
- ENSG00000164251
- UniProt:
- P55085
- OMIM:
- 600933
- Synonyms:
- GPR11, PAR2
Cilia effects upon perturbation of F2RL1
Ciliogenesis screen results (4 screens)
- Kim2016: Not Reported
- Wheway et al. 2015 (siRNA) [siRNA]: Ciliogenesis Defect (z=-4.88) PMID:26167766
- Breslow et al. 2018 (CRISPR) [CRISPR]: No Significant Effect PMID:29459680
- Roosing et al. 2015 (siRNA) [siRNA]: No effect PMID:26595381
Phenotypes
- Mouse phenotype:
- increased startle reflex
Subcellular localization
cilia associated gene, endosome
Functional category
- Ciliary assembly/disassembly
- Trafficking (BBSome, small GTPases, vesicular transport, ATPases)
- Actin & cytoskeleton regulation
- Signaling (Hedgehog, GPCRs, ion channels)
Function
PAR-2 is expressed basolaterally, where it stimulates both intracellular Ca2+ release and Ca2+ influx, which activates low-level nitric oxide production, increases apical membrane Cl− permeability ∼3–5-fold, and increases ciliary beating ∼20–50%( 28874459).